
Substituted conformationally restricted guanidine derivatives: Probing the α2-adrenoceptors' binding pocket
Keywords: Conformationally restricted guanidines; 2-Amino-1,4-dihydroquinazolines; 2-Amino-1,4-dihydropyridopyrimidines; 2-Amino-4,5-dihydro-1,3-benzodiazepines; α2-adrenoceptors' ligands; α2-adrenoceptors' antagonists; Human brain tissue in vitro experiment